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Subject: | | Re: Sinemet and food |
From: | | "Kathrynne Holden, MS, RD" <[log in to unmask]> |
Reply-To: | | PARKINSN: Parkinson's Disease - Information Exchange Network |
Date: | | Tue, 9 Jul 1996 13:41:17 -0400 |
Content-Type: | | text/plain |
Parts/Attachments: |
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Camilla Flintermann wrote:
> I have to confess to some
> confusion about the Sinemet/food connection. We have had very persuasi=
ve
> info from a number of people to the effect that Sinemet taken with food
> loses much of its value by the time it gets out of the stomach. It soun=
ds
> so reasonable--then I notice that Peter's new RX bottle of Sin.CR 50/20=
0
> has a label shouting "TAKE WITH FOOD" !=20
Camilla,
Regular Sinemet is best taken on an empty stomach. Also, protein=20
redistribution may help those who are beginning to experience "on/off"=20
periods. Protein in sizable amounts hinders its absorption; this may not=20
be a problem in early stages of PD, when the brain still produces some=20
dopamine, but may be a problem later on, causing some "freezing" or=20
"off" times. This is because both amino acids (from the protein) and=20
Sinemet require a special carrier to get across across the intestine and=20
into the blood. The aminos and Sinemet compete for these carriers, and=20
if Sinemet is taken with a lot of protein, the aminos win the race.
HOWEVER:
The sustained-release version (Sinemet CR) should be distinguished from=20
Sinemet in this respect. While both contain levodopa/carbidopa=20
combinations, the sustained-release version is designed to work very=20
slowly over a greater period of time, minimizing fluctuations=20
in mobility. It is best taken with food because food takes longer to get=20
through the stomach and intestine; the Sinemet CR goes with it, slowly=20
dissolving along the way.
Here's a paragraph from "Clinical Pharmacology" that may illustrate what=20
I'm saying.
"Pharmacokinetics: Sinemet=AE is administered orally. Following oral=20
administration, amino acid transport mechanisms carry levodopa across=20
the membrane of the GI tract, with approximately 30=9750% of the drug=20
entering the circulation. As a result, high concentrations of amino=20
acids in the GI tract (i.e., a high-protein diet) can interfere with=20
absorption of levodopa. "
As you see, only about 50% of Sinemet makes it out of the intestine and=20
into the blood. Taken with protein, even less Sinemet gets into the=20
blood. But this is not the case with Sinemet CR.
> Now I wonder, are we correct in believing there's a problem, and that w=
e need
> to wait 30-60 min. after taking it before eating?=20
This is true for regular Sinemet.
>Is there something about
> the CR form that makes a difference in this way? =20
As discussed, Sinemet CR should be fine taken with food.
The problem, as I see it, is that for many people, both Sinemet and=20
Sinemet CR must be used. In this case, I'd try to take the Sinemet on an=20
empty stomach, or with carbohydrates, like breads, crackers, etc. Then=20
take the Sin. CR with food.
For a listing of high-protein foods, I'll e-mail the notes I made up on=20
protein distribution separately.
Best regards,
--=20
Kathrynne Holden, MS, RD
Editor-in-Chief,
"Spotlight on Food--nutrition news for people 60-plus"
Tel: 970-493-6532 Fax: 970-493-6538=20
http://www.fortnet.org/~fivstar
You may wish to contact:
Better Business Bureau of the Mountain States,
< [log in to unmask]>
for further information.
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December 1996, Week 3 December 1996, Week 2 December 1996, Week 1 November 1996, Week 5 November 1996, Week 4 November 1996, Week 3 November 1996, Week 2 November 1996, Week 1 October 1996, Week 5 October 1996, Week 4 October 1996, Week 3 October 1996, Week 2 October 1996, Week 1 September 1996, Week 5 September 1996, Week 4 September 1996, Week 3 September 1996, Week 2 September 1996, Week 1 August 1996, Week 5 August 1996, Week 4 August 1996, Week 3 August 1996, Week 2 August 1996, Week 1 July 1996, Week 5 July 1996, Week 4 July 1996, Week 3 July 1996, Week 2 July 1996, Week 1 June 1996, Week 5 June 1996, Week 4 June 1996, Week 3 June 1996, Week 2 June 1996, Week 1 May 1996, Week 5 May 1996, Week 4 May 1996, Week 3 May 1996, Week 2 May 1996, Week 1 April 1996, Week 5 April 1996, Week 4 April 1996, Week 3 April 1996, Week 2 April 1996, Week 1 March 1996, Week 5 March 1996, Week 4 March 1996, Week 3 March 1996, Week 2 March 1996, Week 1 February 1996, Week 5 February 1996, Week 4 February 1996, Week 3 February 1996, Week 2 February 1996, Week 1 January 1996, Week 5 January 1996, Week 4 January 1996, Week 3 January 1996, Week 2 January 1996, Week 1 December 1995, Week 5 December 1995, Week 4 December 1995, Week 3 December 1995, Week 2 December 1995, Week 1 November 1995, Week 5 November 1995, Week 4 November 1995, Week 3 November 1995, Week 2 November 1995, Week 1 October 1995, Week 5 October 1995, Week 4 October 1995, Week 3 October 1995, Week 2 October 1995, Week 1 September 1995, Week 5 September 1995, Week 4 September 1995, Week 3 September 1995, Week 2 September 1995, Week 1 August 1995, Week 5 August 1995, Week 4 August 1995, Week 3 August 1995, Week 2 August 1995, Week 1 July 1995, Week 5 July 1995, Week 4 July 1995, Week 3 July 1995, Week 2 July 1995, Week 1 June 1995, Week 5 June 1995, Week 4 June 1995, Week 3 June 1995, Week 2 June 1995, Week 1 May 1995, Week 5 May 1995, Week 4 May 1995, Week 3 May 1995, Week 2 May 1995, Week 1 April 1995, Week 5 April 1995, Week 4 April 1995, Week 3 April 1995, Week 2 April 1995, Week 1 March 1995, Week 5 March 1995, Week 4 March 1995, Week 3 March 1995, Week 2 March 1995, Week 1 February 1995, Week 4 February 1995, Week 3 February 1995, Week 2 February 1995, Week 1 January 1995, Week 5 January 1995, Week 4 January 1995, Week 3 January 1995, Week 2 January 1995, Week 1 December 1994, Week 5 December 1994, Week 4 December 1994, Week 3 December 1994, Week 2 December 1994, Week 1 November 1994, Week 5 November 1994, Week 4 November 1994, Week 3 November 1994, Week 2 November 1994, Week 1 October 1994, Week 5 October 1994, Week 4 October 1994, Week 3 October 1994, Week 2 October 1994, Week 1 September 1994, Week 5 September 1994, Week 4 September 1994, Week 3 September 1994, Week 2 September 1994, Week 1 August 1994, Week 5 August 1994, Week 4 August 1994, Week 3 August 1994, Week 2 August 1994, Week 1 July 1994, Week 5 July 1994, Week 4 July 1994, Week 3 July 1994, Week 2 July 1994, Week 1 June 1994, Week 5 June 1994, Week 4 June 1994, Week 3 June 1994, Week 2 June 1994, Week 1 May 1994, Week 5 May 1994, Week 4 May 1994, Week 3 May 1994, Week 2 May 1994, Week 1 April 1994, Week 5 April 1994, Week 4 April 1994, Week 3 April 1994, Week 2 April 1994, Week 1 March 1994, Week 5 March 1994, Week 4 March 1994, Week 3 March 1994, Week 2 March 1994, Week 1 February 1994, Week 4 February 1994, Week 3 February 1994, Week 2 February 1994, Week 1 February 1994 January 1994 December 1993 November 1993
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