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PARKINSN Archives
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PARKINSN@LISTSERV.UTORONTO.CA
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Subject: | | Re: drug interaction |
From: | | Margaret Tuchman <[log in to unmask]> |
Reply-To: | | PARKINSN: Parkinson's Disease - Information Exchange Network |
Date: | | Fri, 20 Sep 1996 03:35:59 -0400 |
Content-Type: | | text/plain |
Parts/Attachments: |
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Tina:
As per your request, drug info frm Clinical Pharmacology
PLEASE NOTE:
Levodopa; Carbidopa/Midazolam
Carbidopa-levodopa can cause cardiac arrhythmias if administered before=20
inhalation of hydrocarbon general anesthetics. This interaction is=20
presumably due to the levodopa-induced increases in dopamine.=20
Levodopa-carbidopa should be discontinued 6=978 hours=20
before the administration of general anesthetics.
Patient profile for torrance, tina
Current 4 medications:
=9AAmantadine (Symmetrel=AE)
=9ALevodopa; Carbidopa (Sinemet=AE)=7F
=9AMidazolam (Versed=AE)
=9ASelegiline (Eldepryl=AE)
Drug Interactions Report
Levodopa; Carbidopa/Amantadine
Concomitant administration of amantadine, benztropine, procyclidine, or=20
trihexyphenidyl with levodopa-carbidopa can enhance the therapeutic effec=
ts=20
of levodopa but should not be used in patients with a history of psychosi=
s.
Amantadine can increase the efficiency of levodopa by its action on centr=
al=20
nerve terminals. Patients who exhibit psychoses should avoid this=20
combination because of the possibility of an increased psychotic effect.
Selegiline/Levodopa; Carbidopa
Administration of levodopa to patients receiving drugs that inhibit=20
monoamine oxidase (MAO) can produce a hypertensive response. While=20
traditional MAOIs such as phenelzine inhibit MAO type A and selegiline is=
=20
selective for MAO type B, at doses above 30=9740 mg/day, this selectivity
is lost. Selegiline can increase levodopa-induced dyskinesias, nausea,=20
orthostatic hypotension, confusion, and hallucinations. Reductions in=20
levodopa dosage may be necessary within a few days after the start of=20
selegiline treatment. Even though Parkinson's disease is an indication fo=
r
both selegiline and levodopa, and these 2 drugs are administered together=
=20
safely in some cases, patients should be monitored closely for hypertensi=
ve=20
responses, especially if selegiline doses higher than 10 mg/day are used.=
It=20
is likely, however, that combining selegiline with levodopa-containing=20
products for the treatment of Parkinson's disease may decline due=20
to a report of higher mortality with combination therapy compared to ther=
apy=20
with levodopa without selegiline.=CA=CA=D0=D2
Concomitant use of monoamine oxidase inhibitors (MAOIs) with=20
levodopa-carbidopa can result in hypertensive crisis. Simultaneous use of=
=20
these agents is contraindicated. MAOIs should be discontinued 2=974 weeks=
=20
before initiation of levodopa-carbidopa therapy. Although selegiline
inhibits MOA type B, the adverse effects associated with levodopa, includ=
ing
orthostatic hypotension, confusion, dyskinesias, nausea, and hallucinatio=
ns,=20
can be exacerbated by concomitant administration of selegiline. Dosages o=
f=20
levodopa should be reduced within 2=973 days after beginning selegiline=20
therapy.
Additive Adverse Reactions Report
3 of these drugs may cause:
=95anorexia (amantadine; levodopa/carbidopa; selegiline)
=95nausea/vomiting (amantadine; levodopa/carbidopa; selegiline)
=95orthostatic hypotension (amantadine; levodopa/carbidopa; selegiline)
2 of these drugs may cause:
=95agitation (amantadine; selegiline)
=95anxiety (amantadine; selegiline)
=95ataxia (amantadine; levodopa/carbidopa)
=95confusion (amantadine; selegiline)
=95constipation (amantadine; selegiline)
=95depression (amantadine; selegiline)
=95diarrhea (amantadine; selegiline)
=95dizziness (amantadine; selegiline)
=95drowsiness (amantadine; selegiline)
=95dystonia (levodopa/carbidopa; selegiline)
=95hallucinations (amantadine; selegiline)
=95headache (amantadine; selegiline)
=95hypertension (levodopa/carbidopa; selegiline)
=95insomnia (amantadine; selegiline)
=95neuroleptic malignant syndrome (amantadine; levodopa/carbidopa)=7F
=95urinary retention (levodopa/carbidopa; selegiline)
=95weight loss (levodopa/carbidopa; selegiline)
=95xerostomia (amantadine; selegiline)
Drugs/Contraindications Warning
No potential drug/contraindication warnings were identified.
I wish you good luck.
>i am to have a medical proceedure early tomorrow morning.
>
>the doctor will give me a mild sedative,called FENFANYL
>and/or VERSED.
>
>can anyone tell me if these drugs will interact with my,
>PD meds. I take SINEMET 25/100, ELDEPRYL 5MG,3 AMANTADINE.
Regards,
Margaret Tuchman (54 yrs, dx 1980)
^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^
I've got Parkinson's disease. And he's got mine.
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1998, Week 4 August 1998, Week 3 August 1998, Week 2 August 1998, Week 1 July 1998, Week 5 July 1998, Week 4 July 1998, Week 3 July 1998, Week 2 July 1998, Week 1 June 1998, Week 5 June 1998, Week 4 June 1998, Week 3 June 1998, Week 2 June 1998, Week 1 May 1998, Week 5 May 1998, Week 4 May 1998, Week 3 May 1998, Week 2 May 1998, Week 1 April 1998, Week 5 April 1998, Week 4 April 1998, Week 3 April 1998, Week 2 April 1998, Week 1 March 1998, Week 5 March 1998, Week 4 March 1998, Week 3 March 1998, Week 2 March 1998, Week 1 February 1998, Week 5 February 1998, Week 4 February 1998, Week 3 February 1998, Week 2 February 1998, Week 1 January 1998, Week 5 January 1998, Week 4 January 1998, Week 3 January 1998, Week 2 January 1998, Week 1 December 1997, Week 5 December 1997, Week 4 December 1997, Week 3 December 1997, Week 2 December 1997, Week 1 November 1997, Week 5 November 1997, Week 4 November 1997, Week 3 November 1997, Week 2 November 1997, Week 1 October 1997, Week 5 October 1997, Week 4 October 1997, Week 3 October 1997, Week 2 October 1997, Week 1 September 1997, Week 5 September 1997, Week 4 September 1997, Week 3 September 1997, Week 2 September 1997, Week 1 August 1997, Week 5 August 1997, Week 4 August 1997, Week 3 August 1997, Week 2 August 1997, Week 1 July 1997, Week 5 July 1997, Week 4 July 1997, Week 3 July 1997, Week 2 July 1997, Week 1 June 1997, Week 5 June 1997, Week 4 June 1997, Week 3 June 1997, Week 2 June 1997, Week 1 May 1997, Week 5 May 1997, Week 4 May 1997, Week 3 May 1997, Week 2 May 1997, Week 1 April 1997, Week 5 April 1997, Week 4 April 1997, Week 3 April 1997, Week 2 April 1997, Week 1 March 1997, Week 5 March 1997, Week 4 March 1997, Week 3 March 1997, Week 2 March 1997, Week 1 February 1997, Week 5 February 1997, Week 4 February 1997, Week 3 February 1997, Week 2 February 1997, Week 1 January 1997, Week 5 January 1997, Week 4 January 1997, Week 3 January 1997, Week 2 January 1997, Week 1 December 1996, Week 5 December 1996, Week 4 December 1996, Week 3 December 1996, Week 2 December 1996, Week 1 November 1996, Week 5 November 1996, Week 4 November 1996, Week 3 November 1996, Week 2 November 1996, Week 1 October 1996, Week 5 October 1996, Week 4 October 1996, Week 3 October 1996, Week 2 October 1996, Week 1 September 1996, Week 5 September 1996, Week 4 September 1996, Week 3 September 1996, Week 2 September 1996, Week 1 August 1996, Week 5 August 1996, Week 4 August 1996, Week 3 August 1996, Week 2 August 1996, Week 1 July 1996, Week 5 July 1996, Week 4 July 1996, Week 3 July 1996, Week 2 July 1996, Week 1 June 1996, Week 5 June 1996, Week 4 June 1996, Week 3 June 1996, Week 2 June 1996, Week 1 May 1996, Week 5 May 1996, Week 4 May 1996, Week 3 May 1996, Week 2 May 1996, Week 1 April 1996, Week 5 April 1996, Week 4 April 1996, Week 3 April 1996, Week 2 April 1996, Week 1 March 1996, Week 5 March 1996, Week 4 March 1996, Week 3 March 1996, Week 2 March 1996, Week 1 February 1996, Week 5 February 1996, Week 4 February 1996, Week 3 February 1996, Week 2 February 1996, Week 1 January 1996, Week 5 January 1996, Week 4 January 1996, Week 3 January 1996, Week 2 January 1996, Week 1 December 1995, Week 5 December 1995, Week 4 December 1995, Week 3 December 1995, Week 2 December 1995, Week 1 November 1995, Week 5 November 1995, Week 4 November 1995, Week 3 November 1995, Week 2 November 1995, Week 1 October 1995, Week 5 October 1995, Week 4 October 1995, Week 3 October 1995, Week 2 October 1995, Week 1 September 1995, Week 5 September 1995, Week 4 September 1995, Week 3 September 1995, Week 2 September 1995, Week 1 August 1995, Week 5 August 1995, Week 4 August 1995, Week 3 August 1995, Week 2 August 1995, Week 1 July 1995, Week 5 July 1995, Week 4 July 1995, Week 3 July 1995, Week 2 July 1995, Week 1 June 1995, Week 5 June 1995, Week 4 June 1995, Week 3 June 1995, Week 2 June 1995, Week 1 May 1995, Week 5 May 1995, Week 4 May 1995, Week 3 May 1995, Week 2 May 1995, Week 1 April 1995, Week 5 April 1995, Week 4 April 1995, Week 3 April 1995, Week 2 April 1995, Week 1 March 1995, Week 5 March 1995, Week 4 March 1995, Week 3 March 1995, Week 2 March 1995, Week 1 February 1995, Week 4 February 1995, Week 3 February 1995, Week 2 February 1995, Week 1 January 1995, Week 5 January 1995, Week 4 January 1995, Week 3 January 1995, Week 2 January 1995, Week 1 December 1994, Week 5 December 1994, Week 4 December 1994, Week 3 December 1994, Week 2 December 1994, Week 1 November 1994, Week 5 November 1994, Week 4 November 1994, Week 3 November 1994, Week 2 November 1994, Week 1 October 1994, Week 5 October 1994, Week 4 October 1994, Week 3 October 1994, Week 2 October 1994, Week 1 September 1994, Week 5 September 1994, Week 4 September 1994, Week 3 September 1994, Week 2 September 1994, Week 1 August 1994, Week 5 August 1994, Week 4 August 1994, Week 3 August 1994, Week 2 August 1994, Week 1 July 1994, Week 5 July 1994, Week 4 July 1994, Week 3 July 1994, Week 2 July 1994, Week 1 June 1994, Week 5 June 1994, Week 4 June 1994, Week 3 June 1994, Week 2 June 1994, Week 1 May 1994, Week 5 May 1994, Week 4 May 1994, Week 3 May 1994, Week 2 May 1994, Week 1 April 1994, Week 5 April 1994, Week 4 April 1994, Week 3 April 1994, Week 2 April 1994, Week 1 March 1994, Week 5 March 1994, Week 4 March 1994, Week 3 March 1994, Week 2 March 1994, Week 1 February 1994, Week 4 February 1994, Week 3 February 1994, Week 2 February 1994, Week 1 February 1994 January 1994 December 1993 November 1993
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